Design, Synthesis, and Pharmacological Evaluation of Novel β2/3 Subunit-Selective γ-Aminobutyric Acid Type A (GABA A ) Receptor Modulators

Marco Stadler, Serena Monticelli, Thomas Seidel, Denise Luger, Isabella Salzer, Stefan Boehm, Wolfgang Holzer, Christoph Schwarzer, Ernst Urban, Sophia Khom, Thierry Langer, Vittorio Pace, Steffen Hering

    Publications: Contribution to journalArticlePeer Reviewed

    Original languageEnglish
    Pages (from-to)317-341
    Number of pages25
    JournalJournal of Medicinal Chemistry
    Volume62
    Issue number1
    DOIs
    Publication statusPublished - 1 Oct 2019

    Austrian Fields of Science 2012

    • 301207 Pharmaceutical chemistry
    • 301206 Pharmacology

    Keywords

    • BENZODIAZEPINE BINDING-SITE
    • VALERENIC ACID
    • 3D PHARMACOPHORE
    • INTERNATIONAL UNION
    • EFFICIENT SYNTHESIS
    • LIGAND RECOGNITION
    • NATURAL-PRODUCTS
    • SUBTYPES
    • ANTICONVULSANT
    • CHANNELS

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