Development of new Kir2.1 channel openers from propafenone analogues

Encan Li, Najla Boujeddaine, Marien J.C. Houtman, Renee G.C. Maas, Joost P.G. Sluijter, Gerhard F. Ecker, Anna Stary-Weinzinger, Willem B. van Ham, Marcel A.G. van der Heyden (Corresponding author)

Publications: Contribution to journalArticlePeer Reviewed

Original languageEnglish
Pages (from-to)633-650
Number of pages18
JournalBritish Journal of Pharmacology
Volume182
Issue number3
DOIs
Publication statusPublished - 17 Oct 2024

Austrian Fields of Science 2012

  • 301207 Pharmaceutical chemistry

Keywords

  • cardiac pharmacology
  • drug discovery/target validation
  • hiPSC-CMCs
  • ion channels
  • K2.1 channel
  • off-target effects
  • propafenone analogues

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