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Molecular Insights into hERG Potassium Channel Blockade by Lubeluzole

  • Roberta Gualdani
  • , Maria Maddalena Cavalluzzi
  • , Francesco Tadini-Buoninsegni
  • , Marino Convertino
  • , Philippe Gailly
  • , Anna Stary-Weinzinger
  • , Giovanni Lentini

    Publications: Contribution to journalArticlePeer Reviewed

    Original languageEnglish
    Pages (from-to)2233-2245
    Number of pages13
    JournalCellular Physiology and Biochemistry
    Volume45
    Issue number6
    DOIs
    Publication statusPublished - 2018

    Austrian Fields of Science 2012

    • 301206 Pharmacology

    Keywords

    • Animals
    • CHO Cells
    • Cricetulus
    • Ether-A-Go-Go Potassium Channels/antagonists & inhibitors
    • HEK293 Cells
    • Humans
    • Molecular Docking Simulation
    • Neuroprotective Agents/pharmacology
    • Patch-Clamp Techniques
    • Piperidines/pharmacology
    • Point Mutation
    • Protein Binding
    • Protein Conformation, alpha-Helical
    • Thiazoles/pharmacology
    • DRUG
    • LIGAND EFFICIENCY
    • DETERMINANTS
    • SODIUM-CHANNELS
    • RATS
    • AFFINITY
    • NITRIC-OXIDE
    • INACTIVATED STATE
    • LONG QT SYNDROME
    • hERG channel blockers
    • Patch clamp
    • PHOTOCHEMICAL STROKE MODEL
    • Lubeluzole
    • Ligand efficiency metrics

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