para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

Marco Niello; Daniela Cintulova; Eva Hellsberg; Kathrin Jäntsch; Marion Holy; Leila H. Ayatollahi; Nicholas V. Cozzi; Michael Freissmuth; Walter Sandtner; Gerhard F. Ecker; Marko D. Mihovilovic; Harald H. Sitte

doi:10.1016/j.neuropharm.2019.04.021

para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

Marco Niello, Daniela Cintulova, Eva Hellsberg, Kathrin Jäntsch, Marion Holy, Leila H. Ayatollahi, Nicholas V. Cozzi, Michael Freissmuth, Walter Sandtner, Gerhard F. Ecker, Marko D. Mihovilovic, Harald H. Sitte

Publications: Contribution to journal › Article › Peer Reviewed

Original language	English
Article number	107615
Number of pages	12
Journal	Neuropharmacology
Volume	161
Early online date	24 Apr 2019
DOIs	https://doi.org/10.1016/j.neuropharm.2019.04.021
Publication status	Published - 15 Dec 2019

Austrian Fields of Science 2012

301207 Pharmaceutical chemistry

Keywords

Allosteric
Cathinone
Fluorine
MCAT
Partial-releaser
SERT
RELEASERS
MONOAMINE TRANSPORTERS
DOPAMINE TRANSPORTER
NEUROTRANSMITTER
INTRACRANIAL SELF-STIMULATION
SUBSTRATE
FLUORINE
X-RAY STRUCTURES
LEUT
BINDING

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10.1016/j.neuropharm.2019.04.021

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@article{78bb56f9aec44ee49d6dad8a50046d0e,

title = "para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter",

keywords = "Allosteric, Cathinone, Fluorine, MCAT, Partial-releaser, SERT, RELEASERS, MONOAMINE TRANSPORTERS, DOPAMINE TRANSPORTER, NEUROTRANSMITTER, INTRACRANIAL SELF-STIMULATION, SUBSTRATE, FLUORINE, X-RAY STRUCTURES, LEUT, BINDING",

author = "Marco Niello and Daniela Cintulova and Eva Hellsberg and Kathrin J{\"a}ntsch and Marion Holy and Ayatollahi, {Leila H.} and Cozzi, {Nicholas V.} and Michael Freissmuth and Walter Sandtner and Ecker, {Gerhard F.} and Mihovilovic, {Marko D.} and Sitte, {Harald H.}",

note = "Publisher Copyright: {\textcopyright} 2019",

year = "2019",

month = dec,

day = "15",

doi = "10.1016/j.neuropharm.2019.04.021",

language = "English",

volume = "161",

journal = "Neuropharmacology",

issn = "0028-3908",

}

TY - JOUR

T1 - para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

AU - Niello, Marco

AU - Cintulova, Daniela

AU - Hellsberg, Eva

AU - Jäntsch, Kathrin

AU - Holy, Marion

AU - Ayatollahi, Leila H.

AU - Cozzi, Nicholas V.

AU - Freissmuth, Michael

AU - Sandtner, Walter

AU - Ecker, Gerhard F.

AU - Mihovilovic, Marko D.

AU - Sitte, Harald H.

PY - 2019/12/15

Y1 - 2019/12/15

KW - Allosteric

KW - Cathinone

KW - Fluorine

KW - MCAT

KW - Partial-releaser

KW - SERT

KW - RELEASERS

KW - MONOAMINE TRANSPORTERS

KW - DOPAMINE TRANSPORTER

KW - NEUROTRANSMITTER

KW - INTRACRANIAL SELF-STIMULATION

KW - SUBSTRATE

KW - FLUORINE

KW - X-RAY STRUCTURES

KW - LEUT

KW - BINDING

UR - http://www.scopus.com/inward/record.url?scp=85065525119&partnerID=8YFLogxK

U2 - 10.1016/j.neuropharm.2019.04.021

DO - 10.1016/j.neuropharm.2019.04.021

M3 - Article

C2 - 31028773

AN - SCOPUS:85065525119

SN - 0028-3908

VL - 161

JO - Neuropharmacology

JF - Neuropharmacology

M1 - 107615

ER -

para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

Austrian Fields of Science 2012

Keywords

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Molecular Drug Targets

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para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

Austrian Fields of Science 2012

Keywords

Access to Document

Other files and links

Fingerprint

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Molecular Drug Targets

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