para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

Marco Niello; Daniela Cintulova; Eva Hellsberg; Kathrin Jäntsch; Marion Holy; Leila H. Ayatollahi; Nicholas V. Cozzi; Michael Freissmuth; Walter Sandtner; Gerhard F. Ecker; Marko D. Mihovilovic; Harald H. Sitte

doi:10.1016/j.neuropharm.2019.04.021

para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

Marco Niello
, Daniela Cintulova
, Eva Hellsberg
, Kathrin Jäntsch
, Marion Holy
, Leila H. Ayatollahi
, Nicholas V. Cozzi
, Michael Freissmuth
, Walter Sandtner
, Gerhard F. Ecker
, Marko D. Mihovilovic
, Harald H. Sitte

Publications: Contribution to journal › Article › Peer Reviewed

Original language	English
Article number	107615
Number of pages	12
Journal	Neuropharmacology
Volume	161
Early online date	24 Apr 2019
DOIs	https://doi.org/10.1016/j.neuropharm.2019.04.021
Publication status	Published - 15 Dec 2019

Funding

This work was supported by the Austrian Science Fund/FWF, grant W 1232 ( MolTag) to GFE, MDM and HHS and by the project program grant F35 to GFE and HHS. Appendix A

Austrian Fields of Science 2012

301207 Pharmaceutical chemistry

Keywords

Allosteric
Cathinone
Fluorine
MCAT
Partial-releaser
SERT
RELEASERS
MONOAMINE TRANSPORTERS
DOPAMINE TRANSPORTER
NEUROTRANSMITTER
INTRACRANIAL SELF-STIMULATION
SUBSTRATE
FLUORINE
X-RAY STRUCTURES
LEUT
BINDING

Access to Document

10.1016/j.neuropharm.2019.04.021

Cite this

@article{78bb56f9aec44ee49d6dad8a50046d0e,

title = "para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter",

keywords = "Allosteric, Cathinone, Fluorine, MCAT, Partial-releaser, SERT, RELEASERS, MONOAMINE TRANSPORTERS, DOPAMINE TRANSPORTER, NEUROTRANSMITTER, INTRACRANIAL SELF-STIMULATION, SUBSTRATE, FLUORINE, X-RAY STRUCTURES, LEUT, BINDING",

author = "Marco Niello and Daniela Cintulova and Eva Hellsberg and Kathrin J{\"a}ntsch and Marion Holy and Ayatollahi, \{Leila H.\} and Cozzi, \{Nicholas V.\} and Michael Freissmuth and Walter Sandtner and Ecker, \{Gerhard F.\} and Mihovilovic, \{Marko D.\} and Sitte, \{Harald H.\}",

note = "Publisher Copyright: {\textcopyright} 2019",

year = "2019",

month = dec,

day = "15",

doi = "10.1016/j.neuropharm.2019.04.021",

language = "English",

volume = "161",

journal = "Neuropharmacology",

issn = "0028-3908",

}

TY - JOUR

T1 - para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

AU - Niello, Marco

AU - Cintulova, Daniela

AU - Hellsberg, Eva

AU - Jäntsch, Kathrin

AU - Holy, Marion

AU - Ayatollahi, Leila H.

AU - Cozzi, Nicholas V.

AU - Freissmuth, Michael

AU - Sandtner, Walter

AU - Ecker, Gerhard F.

AU - Mihovilovic, Marko D.

AU - Sitte, Harald H.

PY - 2019/12/15

Y1 - 2019/12/15

KW - Allosteric

KW - Cathinone

KW - Fluorine

KW - MCAT

KW - Partial-releaser

KW - SERT

KW - RELEASERS

KW - MONOAMINE TRANSPORTERS

KW - DOPAMINE TRANSPORTER

KW - NEUROTRANSMITTER

KW - INTRACRANIAL SELF-STIMULATION

KW - SUBSTRATE

KW - FLUORINE

KW - X-RAY STRUCTURES

KW - LEUT

KW - BINDING

UR - https://www.scopus.com/pages/publications/85065525119

U2 - 10.1016/j.neuropharm.2019.04.021

DO - 10.1016/j.neuropharm.2019.04.021

M3 - Article

C2 - 31028773

AN - SCOPUS:85065525119

SN - 0028-3908

VL - 161

JO - Neuropharmacology

JF - Neuropharmacology

M1 - 107615

ER -

para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

Funding

Austrian Fields of Science 2012

Keywords

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Molecular Drug Targets

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para-Trifluoromethyl-methcathinone is an allosteric modulator of the serotonin transporter

Funding

Austrian Fields of Science 2012

Keywords

Access to Document

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Fingerprint

Projects

Molecular Drug Targets

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