Single Peptide Backbone Surrogate Mutations to Regulate Angiotensin GPCR Subtype Selectivity

Eirinaios Vrettos, Ibai E. Valverde, Alba Mascarin, Patrick N. Pallier, Linda Cerofolini, Marco Fragai, Giacomo Parigi, Baydaa Hirmiz, Nick Bekas, Nathalie M. Grob, Hamidreza Shaye, Mark Del Borgo, MarieIsabel Aguilar, Francesca Magnani, Nelofer Syed, Timothy Crook, Emal Waqif, Essam Ghazaly, Vadim Cherezov, Robert E. WiddopClaudio Luchinat, Adina T. MichaelTitus, Thomas L. Mindt (Corresponding author), Andreas G. Tzakos (Corresponding author), Evgenios K. Stylos

Publications: Contribution to journalArticlePeer Reviewed

Original languageEnglish
Pages (from-to)10690-10694
Number of pages5
JournalChemistry: A European Journal
Volume26
Issue number47
DOIs
Publication statusPublished - 21 Aug 2020

Austrian Fields of Science 2012

  • 104026 Spectroscopy
  • 106002 Biochemistry
  • 301305 Medical chemistry

Keywords

  • click chemistry
  • competition-binding experiments
  • G-protein-coupled receptors
  • neurotrophic effects
  • peptidomimetics
  • PEPTIDOMIMETICS

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